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Designing a chemical inhibitor of the AAA protein spastin using active site mutations

Spastin is a microtubule-severing AAA (ATPases associated with diverse cellular activities) protein needed for cell division and intracellular vesicle transport. Currently, we lack chemical inhibitors to probe spastin function in such dynamic cellular processes. To design a chemical inhibitor of spa...

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Dades bibliogràfiques
Publicat a:Nat Chem Biol
Autors principals: Cupido, Tommaso, Pisa, Rudolf, Kelley, Megan E., Kapoor, Tarun M.
Format: Artigo
Idioma:Inglês
Publicat: 2019
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6558985/
https://ncbi.nlm.nih.gov/pubmed/30778202
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41589-019-0225-6
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