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Dual inhibitors of LSD1 and spermine oxidase

We have previously described the synthesis and evaluation of 3,5-diamino-1,2,4-triazole analogues as inhibitors of the flavin-dependent histone demethylase LSD1. These compounds are potent inhibitors of LSD1 without activity against monoamine oxidases A and B, and promote the elevation of H3K4me2 le...

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Pubblicato in:Medchemcomm
Autori principali: Holshouser, Steven, Dunworth, Matthew, Murray-Stewart, Tracy, Peterson, Yuri K., Burger, Pieter, Kirkpatrick, Joy, Chen, Huan-Huan, Casero, Robert A., Woster, Patrick M.
Natura: Artigo
Lingua:Inglês
Pubblicazione: Royal Society of Chemistry 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6533887/
https://ncbi.nlm.nih.gov/pubmed/31191868
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c8md00610e
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