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Dynamic Role of the G Protein in Stabilizing the Active State of the Adenosine A(2A) Receptor

Agonist binding in the extracellular region of the G protein-coupled adenosine A2A receptor increases its affinity to the G proteins in the intracellular region, and vice versa. The structural basis for this effect is not evident from the crystal structures of A(2A)R in various conformational states...

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Bibliographic Details
Published in:Structure
Main Authors: Lee, Sangbae, Nivedha, Anita K., Tate, Christopher G., Vaidehi, Nagarajan
Format: Artigo
Language:Inglês
Published: Cell Press 2019
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Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC6531377/
https://ncbi.nlm.nih.gov/pubmed/30713025
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.str.2018.12.007
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