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Covalent modification of Cys-239 in β-tubulin by small molecules as a strategy to promote tubulin heterodimer degradation

Clinical microtubule-targeting drugs are functionally divided into microtubule-destabilizing and microtubule-stabilizing agents. Drugs from both classes achieve microtubule inhibition by binding different sites on tubulin and inhibiting or promoting polymerization with no concomitant effects on the...

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Dades bibliogràfiques
Publicat a:J Biol Chem
Autors principals: Yang, Jianhong, Li, Yong, Yan, Wei, Li, Weimin, Qiu, Qiang, Ye, Haoyu, Chen, Lijuan
Format: Artigo
Idioma:Inglês
Publicat: American Society for Biochemistry and Molecular Biology 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6527155/
https://ncbi.nlm.nih.gov/pubmed/30940730
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.RA118.006325
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