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Synthesis of deuterium-labelled amlexanox and its metabolic stability against mouse, rat and human microsomes

As part of a program toward making analogues of amlexanox (1), currently under clinical investigation for the treatment of type 2 diabetes and obesity, we have synthesized derivative 5 in which deuterium has been introduced into two sites of metabolism on the C-7 isopropyl function of amlexanox. The...

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Dettagli Bibliografici
Pubblicato in:J Labelled Comp Radiopharm
Autori principali: Gan, Xinmin, Wilson, Michael W., Beyett, Tyler S., Wen, Bo, Sun, Duxin, Larsen, Scott D., Tesmer, John J. G., Saltiel, Alan R., Showalter, Hollis D.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6525014/
https://ncbi.nlm.nih.gov/pubmed/30828860
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/jlcr.3716
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