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Procognitive Properties of Drugs with Single and Multitargeting H(3) Receptor Antagonist Activities

The histamine H(3) receptor (H(3)R) is an important modulator of numerous central control mechanisms. Novel lead optimizations for H(3)R antagonists/inverse agonists involved studies of structure–activity relationships, cross‐affinities, and pharmacokinetic properties of promising ligands. Blockade...

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Bibliografski detalji
Izdano u:CNS Neurosci Ther
Glavni autori: Nikolic, Katarina, Filipic, Slavica, Agbaba, Danica, Stark, Holger
Format: Artigo
Jezik:Inglês
Izdano: John Wiley and Sons Inc. 2014
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6493064/
https://ncbi.nlm.nih.gov/pubmed/24836924
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/cns.12279
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