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Procognitive Properties of Drugs with Single and Multitargeting H(3) Receptor Antagonist Activities

The histamine H(3) receptor (H(3)R) is an important modulator of numerous central control mechanisms. Novel lead optimizations for H(3)R antagonists/inverse agonists involved studies of structure–activity relationships, cross‐affinities, and pharmacokinetic properties of promising ligands. Blockade...

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Bibliographic Details
Published in:CNS Neurosci Ther
Main Authors: Nikolic, Katarina, Filipic, Slavica, Agbaba, Danica, Stark, Holger
Format: Artigo
Language:Inglês
Published: John Wiley and Sons Inc. 2014
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC6493064/
https://ncbi.nlm.nih.gov/pubmed/24836924
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/cns.12279
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