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Procognitive Properties of Drugs with Single and Multitargeting H(3) Receptor Antagonist Activities
The histamine H(3) receptor (H(3)R) is an important modulator of numerous central control mechanisms. Novel lead optimizations for H(3)R antagonists/inverse agonists involved studies of structure–activity relationships, cross‐affinities, and pharmacokinetic properties of promising ligands. Blockade...
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| Publicado no: | CNS Neurosci Ther |
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| Main Authors: | , , , |
| Formato: | Artigo |
| Idioma: | Inglês |
| Publicado em: |
John Wiley and Sons Inc.
2014
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| Assuntos: | |
| Acesso em linha: | https://ncbi.nlm.nih.gov/pmc/articles/PMC6493064/ https://ncbi.nlm.nih.gov/pubmed/24836924 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/cns.12279 |
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