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Procognitive Properties of Drugs with Single and Multitargeting H(3) Receptor Antagonist Activities

The histamine H(3) receptor (H(3)R) is an important modulator of numerous central control mechanisms. Novel lead optimizations for H(3)R antagonists/inverse agonists involved studies of structure–activity relationships, cross‐affinities, and pharmacokinetic properties of promising ligands. Blockade...

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Detalhes bibliográficos
Publicado no:CNS Neurosci Ther
Main Authors: Nikolic, Katarina, Filipic, Slavica, Agbaba, Danica, Stark, Holger
Formato: Artigo
Idioma:Inglês
Publicado em: John Wiley and Sons Inc. 2014
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6493064/
https://ncbi.nlm.nih.gov/pubmed/24836924
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/cns.12279
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