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Procognitive Properties of Drugs with Single and Multitargeting H(3) Receptor Antagonist Activities

The histamine H(3) receptor (H(3)R) is an important modulator of numerous central control mechanisms. Novel lead optimizations for H(3)R antagonists/inverse agonists involved studies of structure–activity relationships, cross‐affinities, and pharmacokinetic properties of promising ligands. Blockade...

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Détails bibliographiques
Publié dans:CNS Neurosci Ther
Auteurs principaux: Nikolic, Katarina, Filipic, Slavica, Agbaba, Danica, Stark, Holger
Format: Artigo
Langue:Inglês
Publié: John Wiley and Sons Inc. 2014
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC6493064/
https://ncbi.nlm.nih.gov/pubmed/24836924
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/cns.12279
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