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Novel 8-Substituted Coumarins That Selectively Inhibit Human Carbonic Anhydrase IX and XII

A novel series of 8-substituted coumarin-based compounds, characterized by the presence of alkylpiperazine and arylpiperazine chains, were synthesized and tested for their inhibitory activity against four human carbonic anhydrase (hCA) isoforms. All compounds displayed nanomolar potency against the...

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Detalles Bibliográficos
Publicado en:Int J Mol Sci
Autores principales: Buran, Kerem, Bua, Silvia, Poli, Giulio, Önen Bayram, F. Esra, Tuccinardi, Tiziano, T. Supuran, Claudiu
Formato: Artigo
Lenguaje:Inglês
Publicado: MDPI 2019
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6429297/
https://ncbi.nlm.nih.gov/pubmed/30857344
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms20051208
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