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Catalytic β C–H amination via an imidate radical relay

The first catalytic strategy to harness imidate radicals for C–H functionalization has been developed. This iodine-catalyzed approach enables β C–H amination of alcohols by an imidate-mediated radical relay. In contrast to our first-generation, (super)stoichiometric protocol, this catalytic method e...

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Detalhes bibliográficos
Publicado no:Chem Sci
Main Authors: Stateman, Leah M., Wappes, Ethan A., Nakafuku, Kohki M., Edwards, Kara M., Nagib, David A.
Formato: Artigo
Idioma:Inglês
Publicado em: Royal Society of Chemistry 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6419930/
https://ncbi.nlm.nih.gov/pubmed/30996986
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c8sc05685d
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