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Development of matrix metalloproteinase-13 inhibitors – A structure-activity/structure-property relationship study

A structure-activity/structure-property relationship study based on the physicochemical as well as in vitro pharmacokinetic properties of a first generation matrix metalloproteinase (MMP)-13 inhibitor (2) was undertaken. After systematic variation of inhibitor 2, compound 31 was identified which exh...

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Détails bibliographiques
Publié dans:Bioorg Med Chem
Auteurs principaux: Fuerst, Rita, Choi, Jun Yong, Knapinska, Anna M., Smith, Lyndsay, Cameron, Michael D., Ruiz, Claudia, Fields, Gregg B., Roush, William R.
Format: Artigo
Langue:Inglês
Publié: 2018
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC6379921/
https://ncbi.nlm.nih.gov/pubmed/30249495
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2018.08.020
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