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Tetrahydroisoquinoline Sulfamates as Potent Microtubule Disruptors: Synthesis, Antiproliferative and Antitubulin Activity of Dichlorobenzyl-Based Derivatives, and a Tubulin Cocrystal Structure

[Image: see text] Tetrahydroisoquinoline (THIQ) 6-O-sulfamate-based anticancer agents, inspired by the endogenous steroid 2-methoxyestradiol and its sulfamate derivatives, are further explored for antiproliferative and microtubule disruptor activity. Based on recently designed C3-methyl C7-methoxy-s...

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Bibliografiske detaljer
Udgivet i:ACS Omega
Main Authors: Dohle, Wolfgang, Prota, Andrea E., Menchon, Grégory, Hamel, Ernest, Steinmetz, Michel O., Potter, Barry V. L.
Format: Artigo
Sprog:Inglês
Udgivet: American Chemical Society 2019
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6372245/
https://ncbi.nlm.nih.gov/pubmed/30775645
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsomega.8b02879
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