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Development of potent pyrazolopyrimidinone-based WEE1 inhibitors with limited single-agent cytotoxicity for cancer therapy

WEE1 kinase regulates the G2-M cell-cycle checkpoint, a critical mechanism for DNA repair in cancer cells that can confer resistance to DNA-damaging agents. We previously reported a series of pyrazolopyrimidinones based on AZD1775, a known WEE1 inhibitor, as an initial investigation into the structu...

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Detalhes bibliográficos
Publicado no:ChemMedChem
Main Authors: Matheson, Christopher J., Casalvieri, Kimberly A, Backos, Donald S., Reigan, Philip
Formato: Artigo
Idioma:Inglês
Publicado em: 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6370589/
https://ncbi.nlm.nih.gov/pubmed/29883531
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.201800188
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