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Mitogen-Activated Protein Kinase Signaling Mediates Opioid-induced Presynaptic NMDA Receptor Activation and Analgesic Tolerance

Opioid-induced hyperalgesia and analgesic tolerance can lead to dose escalation and inadequate pain treatment with μ-opioid receptor agonists. Opioids cause tonic activation of glutamate NMDA receptors (NMDARs) at primary afferent terminals, increasing nociceptive input. However, the signaling mecha...

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Detalhes bibliográficos
Publicado no:J Neurochem
Main Authors: Deng, Meichun, Chen, Shao-Rui, Chen, Hong, Luo, Yi, Dong, Yingchun, Pan, Hui-Lin
Formato: Artigo
Idioma:Inglês
Publicado em: 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6340739/
https://ncbi.nlm.nih.gov/pubmed/30444263
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/jnc.14628
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