Cargando...

Small Molecule Targeting of Protein–Protein Interactions through Allosteric Modulation of Dynamics

The protein–protein interaction (PPI) target class is particularly challenging, but offers potential for “first in class” therapies. Most known PPI small molecules are orthosteric inhibitors but many PPI sites may be fundamentally intractable to this approach. One potential alternative is to conside...

Descripción completa

Guardado en:
Detalles Bibliográficos
Publicado en:Molecules
Autores principales: Cossins, Benjamin P., Lawson, Alastair D. G.
Formato: Artigo
Lenguaje:Inglês
Publicado: MDPI 2015
Materias:
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6332300/
https://ncbi.nlm.nih.gov/pubmed/26378508
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules200916435
Etiquetas: Agregar Etiqueta
Sin Etiquetas, Sea el primero en etiquetar este registro!