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Targeting epigenetic protein–protein interactions with small-molecule inhibitors

Epigenetic protein–protein interactions (PPIs) play essential roles in regulating gene expression, and their dysregulations have been implicated in many diseases. These PPIs are comprised of reader domains recognizing post-translational modifications on histone proteins, and of scaffolding proteins...

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Detalhes bibliográficos
Publicado no:Future Med Chem
Main Authors: Linhares, Brian M, Grembecka, Jolanta, Cierpicki, Tomasz
Formato: Artigo
Idioma:Inglês
Publicado em: Newlands Press Ltd 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7421387/
https://ncbi.nlm.nih.gov/pubmed/32551894
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.4155/fmc-2020-0082
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