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Targeting epigenetic protein–protein interactions with small-molecule inhibitors

Epigenetic protein–protein interactions (PPIs) play essential roles in regulating gene expression, and their dysregulations have been implicated in many diseases. These PPIs are comprised of reader domains recognizing post-translational modifications on histone proteins, and of scaffolding proteins...

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Kaydedildi:
Detaylı Bibliyografya
Yayımlandı:Future Med Chem
Asıl Yazarlar: Linhares, Brian M, Grembecka, Jolanta, Cierpicki, Tomasz
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: Newlands Press Ltd 2020
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC7421387/
https://ncbi.nlm.nih.gov/pubmed/32551894
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.4155/fmc-2020-0082
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