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Differential PROTAC substrate specificity dictated by orientation of recruited E3 ligase

PROteolysis-TArgeting Chimeras (PROTACs) are hetero-bifunctional molecules that recruit an E3 ubiquitin ligase to a given substrate protein resulting in its targeted degradation. Many potent PROTACs with specificity for dissimilar targets have been developed; however, the factors governing degradati...

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Bibliografiset tiedot
Julkaisussa:Nat Commun
Päätekijät: Smith, Blake E., Wang, Stephen L., Jaime-Figueroa, Saul, Harbin, Alicia, Wang, Jing, Hamman, Brian D., Crews, Craig M.
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: Nature Publishing Group UK 2019
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC6328587/
https://ncbi.nlm.nih.gov/pubmed/30631068
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41467-018-08027-7
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