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Synthesis of aminopyrazole analogs and their evaluation as CDK inhibitors for cancer therapy

We synthesized a library of aminopyrazole analogs to systematically explore the hydrophobic pocket adjacent to the hinge region and the solvent exposed region of cyclin dependent kinases. Structure-activity relationship studies identified an optimal substitution in the hydrophobic pocket and analog...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem Lett
Main Authors: Rana, Sandeep, Sonawane, Yogesh A., Taylor, Margaret A., Kizhake, Smitha, Zahid, Muhammad, Natarajan, Amarnath
Formato: Artigo
Idioma:Inglês
Publicado em: 2018
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6295223/
https://ncbi.nlm.nih.gov/pubmed/30343954
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2018.10.020
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