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Several structural motifs cooperate in determining the highly effective anti-thrombin activity of NU172 aptamer

Despite aptamers are very promising alternative to antibodies, very few of them are under clinical trials or are used as drugs. Among them, NU172 is currently in Phase II as anticoagulant in heart disease treatments. It inhibits thrombin activity much more effectively than TBA, the best-known thromb...

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Dades bibliogràfiques
Publicat a:Nucleic Acids Res
Autors principals: Troisi, Romualdo, Napolitano, Valeria, Spiridonova, Vera, Russo Krauss, Irene, Sica, Filomena
Format: Artigo
Idioma:Inglês
Publicat: Oxford University Press 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6294562/
https://ncbi.nlm.nih.gov/pubmed/30357392
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/nar/gky990
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