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Si-Directed regiocontrol in asymmetric Pd-catalyzed allylic alkylations using C1-ammonium enolate nucleophiles

Cooperative catalysis enables the direct enantioselective α-allylation of linear prochiral esters using Si-substituted allyl electrophiles. The Si-substituent directs the regioselectivity of enantioselective bond formation and provides products containing synthetically versatile pentafluorophenyl es...

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Publicado en:Tetrahedron
Autores principales: Fyfe, James W. B., Kabia, Omaru M., Pearson, Colin M., Snaddon, Thomas N.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2018
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6294469/
https://ncbi.nlm.nih.gov/pubmed/30559533
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.tet.2018.04.021
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