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Design of novel lipidated peptidomimetic conjugates for targeting EGFR heterodimerization in HER2 + cancer

The human epidermal growth factor receptor (EGFR) family is known to be involved in cell signaling pathways. The extracellular domain of EGFR consists of four domains, of which domain II and domain IV are known to be involved in the dimerization process. Overexpression of these receptors is known to...

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Publicat a:Bioorg Med Chem Lett
Autors principals: Naik, Himgauri, Gauthier, Ted, Singh, Sitanshu, Jois, Seetharama
Format: Artigo
Idioma:Inglês
Publicat: 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6283100/
https://ncbi.nlm.nih.gov/pubmed/30314880
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2018.10.005
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