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Lead Discovery of Type II BRAF V600E Inhibitors Targeting the Structurally Validated DFG-Out Conformation Based upon Selected Fragments

The success of the first approved kinase inhibitor imatinib has spurred great interest in the development of type II inhibitors targeting the inactive DFG-out conformation, wherein the Phe of the DFG motif at the start of the activation loop points into the ATP binding site. Nevertheless, kinase inh...

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Detalhes bibliográficos
Publicado no:Molecules
Main Authors: Zhang, Qingwen, Zhang, Xuejin, You, Qidong
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6272942/
https://ncbi.nlm.nih.gov/pubmed/27438814
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules21070879
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