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Design, Synthesis and Anti-fibrosis Activity Study of N(1)-Substituted Phenylhydroquinolinone Derivatives
Pirfenidone (5-methyl-1-phenyl-2(1H)-pyridone, PFD) is a small-molecule compound acting on multiple targets involved in pathological fibrogenesis and is effective to increase the survival of patients with fibrosis, such as idiopathic pulmonary fibrosis. However, PFD is not active enough, requiring a...
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| Publicado en: | Molecules |
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| Autores principales: | , , , , , |
| Formato: | Artigo |
| Lenguaje: | Inglês |
| Publicado: |
MDPI
2012
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| Materias: | |
| Acceso en línea: | https://ncbi.nlm.nih.gov/pmc/articles/PMC6269057/ https://ncbi.nlm.nih.gov/pubmed/22301723 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules17021373 |
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