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Chemistry and Structure-Activity Relationship of the Styrylquinoline-Type HIV Integrase Inhibitors

In spite of significant progress in anti-HIV-1 therapy, current antiviral chemo-therapy still suffers from deleterious side effects and emerging drug resistance. Therefore, the development of novel antiviral drugs remains a crucial issue for the fight against AIDS. HIV-1 integrase is a key enzyme in...

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Publicado no:Molecules
Main Authors: Mouscadet, Jean-François, Desmaële, Didier
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6263292/
https://ncbi.nlm.nih.gov/pubmed/20657464
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules15053048
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