A carregar...

Affinity, potency, efficacy, and selectivity of neurokinin A analogs at human recombinant NK2 and NK1 receptors

A series of peptide NK2 receptor agonists was evaluated for affinity, potency, efficacy, and selectivity at human recombinant NK2 and NK1 receptors expressed in CHO cells to identify compounds with the greatest separation between NK2 and NK1 receptor agonist activity. Binding studies were performed...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Publicado no:PLoS One
Main Authors: Rupniak, Nadia M. J., Perdona, Elisabetta, Griffante, Cristiana, Cavallini, Palmina, Sava, Anna, Ricca, Daniel J., Thor, Karl B., Burgard, Edward C., Corsi, Mauro
Formato: Artigo
Idioma:Inglês
Publicado em: Public Library of Science 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6201908/
https://ncbi.nlm.nih.gov/pubmed/30359406
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0205894
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!