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[(3)H]GR205171 displays similar NK1 receptor binding profile in gerbil and human brain

1. In this study, [(3)H]GR205171 (3(S)-(2-methoxy-5-(5-trifluoromethyltetrazol-1-yl)-phenylmethylamino)-2(S)-phenylpiperidine), a potent and selective NK1 receptor antagonist, was characterised in autoradiographic studies in gerbil brain and in binding experiments on homogenates from gerbil and huma...

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Autors principals: Griffante, Cristiana, Carletti, Renzo, Andreetta, Filippo, Corsi, Mauro
Format: Artigo
Idioma:Inglês
Publicat: Nature Publishing Group 2006
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC1617048/
https://ncbi.nlm.nih.gov/pubmed/16501582
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0706697
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