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Small-molecule TLR8 antagonists via structure-based rational design

Rational design of drug-like small-molecule ligands based on structural information of proteins remains a significant challenge in chemical biology. In particular, designs targeting protein-protein interfaces have met little success given the dynamic nature of the protein surfaces. Herein, we utiliz...

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Detalhes bibliográficos
Publicado no:Cell Chem Biol
Main Authors: Hu, Zhenyi, Tanji, Hiromi, Jiang, Shuangshuang, Zhang, Shuting, Koo, Kyoin, Chan, Jean, Sakaniwa, Kentaro, Ohto, Umeharu, Candia, Albert, Shimizu, Toshiyuki, Yin, Hang
Formato: Artigo
Idioma:Inglês
Publicado em: 2018
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6195466/
https://ncbi.nlm.nih.gov/pubmed/30100350
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2018.07.004
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