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Quantitative Structure–Activity Relationship Modeling of Kinase Selectivity Profiles

The discovery of selective inhibitors of biological target proteins is the primary goal of many drug discovery campaigns. However, this goal has proven elusive, especially for inhibitors targeting the well-conserved orthosteric adenosine triphosphate (ATP) binding pocket of kinase enzymes. The human...

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Détails bibliographiques
Publié dans:Molecules
Auteurs principaux: Kothiwale, Sandeepkumar, Borza, Corina, Pozzi, Ambra, Meiler, Jens
Format: Artigo
Langue:Inglês
Publié: MDPI 2017
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC6151389/
https://ncbi.nlm.nih.gov/pubmed/28925954
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules22091576
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