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Discoidin domain receptor 1 (DDR1) kinase as target for structure-based drug discovery

Discoidin domain receptor (DDR) 1 and 2 are transmembrane receptors that belong to the family of receptor tyrosine kinases (RTK). Upon collagen binding, DDRs transduce cellular signaling involved in various cell functions, including cell adhesion, proliferation, differentiation, migration, and matri...

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Dettagli Bibliografici
Pubblicato in:Drug Discov Today
Autori principali: Kothiwale, Sandeepkumar, Borza, Corina M., Lowe, Will, Pozzi, Ambra, Meiler, Jens
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2014
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4336622/
https://ncbi.nlm.nih.gov/pubmed/25284748
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.drudis.2014.09.025
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