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Discoidin domain receptor 1 (DDR1) kinase as target for structure-based drug discovery

Discoidin domain receptor (DDR) 1 and 2 are transmembrane receptors that belong to the family of receptor tyrosine kinases (RTK). Upon collagen binding, DDRs transduce cellular signaling involved in various cell functions, including cell adhesion, proliferation, differentiation, migration, and matri...

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Podrobná bibliografie
Vydáno v:Drug Discov Today
Hlavní autoři: Kothiwale, Sandeepkumar, Borza, Corina M., Lowe, Will, Pozzi, Ambra, Meiler, Jens
Médium: Artigo
Jazyk:Inglês
Vydáno: 2014
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4336622/
https://ncbi.nlm.nih.gov/pubmed/25284748
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.drudis.2014.09.025
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