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Targeting kinases with precision

Cancer genomics and mechanistic studies have revealed that heterogeneous mutations within a single kinase can result in a variety of activation mechanisms. The challenge has been to match these insights with tailored drug discovery strategies to yield potent, highly selective drugs. With optimized d...

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Dettagli Bibliografici
Pubblicato in:Mol Cell Oncol
Autori principali: Gardino, Alexandra K., Evans, Erica K., Kim, Joseph L., Brooijmans, Natasja, Hodous, Brian L., Wolf, Beni, Lengauer, Christoph
Natura: Artigo
Lingua:Inglês
Pubblicazione: Taylor & Francis 2018
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6149809/
https://ncbi.nlm.nih.gov/pubmed/30250891
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/23723556.2018.1435183
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