Wordt geladen...

Virtual screening using covalent docking to find activators for G245S mutant p53

TP53 is the most mutated gene in all cancers. The mutant protein also accumulates in cells. The high frequency of p53 mutations makes the protein a promising target for anti-cancer therapy. Only a few molecules have been found, using in vitro screening, to reactivate the mutant protein. APR-246 is c...

Volledige beschrijving

Bewaard in:
Bibliografische gegevens
Gepubliceerd in:PLoS One
Hoofdauteurs: Omar, Sara Ibrahim, Lepre, Marco Gaetano, Morbiducci, Umberto, Deriu, Marco Agostino, Tuszynski, Jack A.
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: Public Library of Science 2018
Onderwerpen:
Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6128461/
https://ncbi.nlm.nih.gov/pubmed/30192754
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0200769
Tags: Voeg label toe
Geen labels, Wees de eerste die dit record labelt!