Wird geladen...

Novel valdecoxib derivatives by ruthenium(ii)-promoted 1,3-dipolar cycloaddition of nitrile oxides with alkynes – synthesis and COX-2 inhibition activity

Novel valdecoxib-based cyclooxygenase-2 inhibitors were synthesized in one step via 1,3-dipolar cycloaddition of nitrile oxides with a series of eleven aryl alkynes, six of them described for the first time. Application of Ru(ii)-catalysis leads preferably to the formation of the 3,4-diaryl-substitu...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Veröffentlicht in:Medchemcomm
Hauptverfasser: Roscales, Silvia, Bechmann, Nicole, Weiss, Daniel Holger, Köckerling, Martin, Pietzsch, Jens, Kniess, Torsten
Format: Artigo
Sprache:Inglês
Veröffentlicht: Royal Society of Chemistry 2018
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6072335/
https://ncbi.nlm.nih.gov/pubmed/30108944
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c7md00575j
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!