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Assessment of Substrate-Dependent Ligand Interactions at the Organic Cation Transporter OCT2 Using Six Model Substrates

Organic cation transporter (OCT) 2 mediates the entry step for organic cation secretion by renal proximal tubule cells and is a site of unwanted drug-drug interactions (DDIs). But reliance on decision tree–based predictions of DDIs at OCT2 that depend on IC(50) values can be suspect because they can...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Veröffentlicht in:Mol Pharmacol
Hauptverfasser: Sandoval, Philip J., Zorn, Kimberley M., Clark, Alex M., Ekins, Sean, Wright, Stephen H.
Format: Artigo
Sprache:Inglês
Veröffentlicht: The American Society for Pharmacology and Experimental Therapeutics 2018
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6070079/
https://ncbi.nlm.nih.gov/pubmed/29884691
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.117.111443
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