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Structural basis for selective inhibition of human PKG Iα by the balanol-like compound N46

Activation of protein kinase G (PKG) Iα in nociceptive neurons induces long-term hyperexcitability that causes chronic pain. Recently, a derivative of the fungal metabolite balanol, N46, has been reported to inhibit PKG Iα with high potency and selectivity and attenuate thermal hyperalgesia and oste...

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Bibliografski detalji
Izdano u:J Biol Chem
Glavni autori: Qin, Liying, Sankaran, Banumathi, Aminzai, Sahar, Casteel, Darren E., Kim, Choel
Format: Artigo
Jezik:Inglês
Izdano: American Society for Biochemistry and Molecular Biology 2018
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6052212/
https://ncbi.nlm.nih.gov/pubmed/29769318
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.RA118.002427
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