Synthesis of novel benzenesulfamide derivatives with inhibitory activity against human cytosolic carbonic anhydrase I and II and Vibrio cholerae α- and β-class enzymes

The synthesis of a new series of sulfamides incorporating ortho-, meta, and para-benzenesulfamide moieties is reported, which were investigated for the inhibition of two human (h) isoforms of the zinc enzyme carbonic anhydrase (CA, EC 4.2.1.1), hCA I and II, and two Vibrio cholerae enzymes, belongin...

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Detalhes bibliográficos
Publicado no:J Enzyme Inhib Med Chem
Main Authors: Bua, Silvia, Berrino, Emanuela, Del Prete, Sonia, Murthy, Vallabhaneni S., Vijayakumar, Vijayaparthasarathi, Tamboli, Yasinalli, Capasso, Clemente, Cerbai, Elisabetta, Mugelli, Alessandro, Carta, Fabrizio, Supuran, Claudiu T.
Formato: Artigo
Idioma:Inglês
Publicado em: Taylor & Francis 2018
Assuntos:
Research Paper
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6041819/
https://ncbi.nlm.nih.gov/pubmed/29987956
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/14756366.2018.1467901
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