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Zinc Metallochaperones as Mutant p53 Reactivators: A New Paradigm in Cancer Therapeutics

Restoration of wild-type structure and function to mutant p53 with a small molecule (hereafter referred to as “reactivating” mutant p53) is one of the holy grails in cancer therapeutics. The majority of TP53 mutations are missense which generate a defective protein that is targetable. We are current...

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Dettagli Bibliografici
Pubblicato in:Cancers (Basel)
Autori principali: Kogan, Samuel, Carpizo, Darren R.
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6025018/
https://ncbi.nlm.nih.gov/pubmed/29843463
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/cancers10060166
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