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HIV anti-latency treatment mediated by macromolecular prodrugs of histone deacetylase inhibitor, panobinostat

Histone deacetylase inhibitors (HDACi) and panobinostat in particular are currently in the focus of intensive investigation as latency reversing agents against the human immunodeficiency virus (HIV). Regretfully, HDACi have dose limiting side-effects making controlled, optimized methods for delivery...

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Vydáno v:Chem Sci
Hlavní autoři: Zuwala, Kaja, Smith, Anton A. A., Tolstrup, Martin, Zelikin, Alexander N.
Médium: Artigo
Jazyk:Inglês
Vydáno: Royal Society of Chemistry 2016
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6003675/
https://ncbi.nlm.nih.gov/pubmed/29997778
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c5sc03257a
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