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Polypharmacology Within the Full Kinome: a Machine Learning Approach

Protein kinases generate nearly a thousand different protein products and regulate the majority of cellular pathways and signal transduction. It is therefore not surprising that the deregulation of kinases has been implicated in many disease states. In fact, kinase inhibitors are the largest class o...

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Publicat a:AMIA Jt Summits Transl Sci Proc
Autors principals: Jones, Derek, Bopaiah, Jeevith, Alghamedy, Fatemah, Jacobs, Nathan, Weiss, Heidi L., de Jong, W.A., Ellingson, Sally R.
Format: Artigo
Idioma:Inglês
Publicat: American Medical Informatics Association 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5961802/
https://ncbi.nlm.nih.gov/pubmed/29888050
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