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Synthesis and biological evaluation of stilbene analogs as Hsp90 C-terminal inhibitors

The design, synthesis and biological evaluation of stilbene-based novobiocin analogs is reported. Replacement of the biaryl amide side chain with a triazole side chain produced compounds that exhibited good anti-proliferative activities. Hsp90 inhibition was observed when N-methyl piperidine was rep...

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Publicado en:ChemMedChem
Autores principales: Byrd, Katherine M., Kent, Caitlin N., Blagg, Brian S. J.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2017
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5892432/
https://ncbi.nlm.nih.gov/pubmed/29058824
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.201700630
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