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Design, Synthesis, and Biological Evaluation of Ring-Constrained Novobiocin Analogues as Hsp90 C-Terminal Inhibitors

[Image: see text] Hsp90 C-terminal inhibitors represent a novel and alternative chemotherapeutic approach for the treatment of cancer. Novobiocin was the first natural product identified as an Hsp90 C-terminal inhibitor; however, it manifests poor antiproliferative activity. In contrast to N-termina...

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Detalles Bibliográficos
Publicado en:ACS Med Chem Lett
Main Authors: Garg, Gaurav, Zhao, Huiping, Blagg, Brian S. J.
Formato: Artigo
Idioma:Inglês
Publicado: American Chemical Society 2014
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4329597/
https://ncbi.nlm.nih.gov/pubmed/25699150
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml5004475
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