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Orally Disintegrating Tablets Containing Melt Extruded Amorphous Solid Dispersion of Tacrolimus for Dissolution Enhancement

In order to improve the aqueous solubility and dissolution of Tacrolimus (TAC), amorphous solid dispersions of TAC were prepared by hot melt extrusion with three hydrophilic polymers, Polyvinylpyrrolidone vinyl acetate (PVP VA64), Soluplus(®) and Hydroxypropyl Cellulose (HPC), at a drug loading of 1...

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Detalhes bibliográficos
Publicado no:Pharmaceutics
Main Authors: Ponnammal, Poovizhi, Kanaujia, Parijat, Yani, Yin, Ng, Wai Kiong, Tan, Reginald B. H.
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5874848/
https://ncbi.nlm.nih.gov/pubmed/29547585
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics10010035
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