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Design, synthesis, and in vitro evaluation of quinolinyl analogues for α-synuclein aggregation

Here we report the synthesis and in vitro evaluation of 25 new quinolinyl analogues for α-synuclein aggregates. Three lead compounds were subsequently labeled with carbon-11 or fluorine-18 to directly assess their potency in a direct radioactive competitive binding assay ng both α-synuclein fibrils...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem Lett
Main Authors: Yue, Xuyi, Dhavale, Dhruva D., Li, Junfeng, Luo, Zonghua, Liu, Jialu, Yang, Hao, Mach, Robert H., Kotzbauer, Paul T., Tu, Zhude
Formato: Artigo
Idioma:Inglês
Publicado em: 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5870887/
https://ncbi.nlm.nih.gov/pubmed/29482941
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2018.02.031
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