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Molecular recognition of ternary complexes: a new dimension in the structure-guided design of chemical degraders

Molecular glues and bivalent inducers of protein degradation (also known as PROTACs) represent a fascinating new modality in pharmacotherapeutics: the potential to knockdown previously thought ‘undruggable’ targets at sub-stoichiometric concentrations in ways not possible using conventional inhibito...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Essays Biochem
Egile Nagusiak: Hughes, Scott J., Ciulli, Alessio
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Portland Press Ltd. 2017
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC5869862/
https://ncbi.nlm.nih.gov/pubmed/29118097
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1042/EBC20170041
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