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Predict drug permeability to blood–brain-barrier from clinical phenotypes: drug side effects and drug indications

Motivation: Blood–Brain-Barrier (BBB) is a rigorous permeability barrier for maintaining homeostasis of Central Nervous System (CNS). Determination of compound’s permeability to BBB is prerequisite in CNS drug discovery. Existing computational methods usually predict drug BBB permeability from chemi...

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Dettagli Bibliografici
Pubblicato in:Bioinformatics
Autori principali: Gao, Zhen, Chen, Yang, Cai, Xiaoshu, Xu, Rong
Natura: Artigo
Lingua:Inglês
Pubblicazione: Oxford University Press 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5860495/
https://ncbi.nlm.nih.gov/pubmed/27993785
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/bioinformatics/btw713
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