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Predict drug permeability to blood–brain-barrier from clinical phenotypes: drug side effects and drug indications

Motivation: Blood–Brain-Barrier (BBB) is a rigorous permeability barrier for maintaining homeostasis of Central Nervous System (CNS). Determination of compound’s permeability to BBB is prerequisite in CNS drug discovery. Existing computational methods usually predict drug BBB permeability from chemi...

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Bibliografski detalji
Izdano u:Bioinformatics
Glavni autori: Gao, Zhen, Chen, Yang, Cai, Xiaoshu, Xu, Rong
Format: Artigo
Jezik:Inglês
Izdano: Oxford University Press 2017
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC5860495/
https://ncbi.nlm.nih.gov/pubmed/27993785
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/bioinformatics/btw713
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