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Predict drug permeability to blood–brain-barrier from clinical phenotypes: drug side effects and drug indications

Motivation: Blood–Brain-Barrier (BBB) is a rigorous permeability barrier for maintaining homeostasis of Central Nervous System (CNS). Determination of compound’s permeability to BBB is prerequisite in CNS drug discovery. Existing computational methods usually predict drug BBB permeability from chemi...

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Detalhes bibliográficos
Publicado no:Bioinformatics
Main Authors: Gao, Zhen, Chen, Yang, Cai, Xiaoshu, Xu, Rong
Formato: Artigo
Idioma:Inglês
Publicado em: Oxford University Press 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5860495/
https://ncbi.nlm.nih.gov/pubmed/27993785
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/bioinformatics/btw713
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