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Synthesis and Evaluation of Pyridyloxypyridyl Indole Carboxamides as Potential PET Imaging Agents for 5-HT(2C) Receptors

[Image: see text] Nine pyridyloxypyridyl indole carboxamides were synthesized and displayed high affinities for 5-HT(2C) receptors and high selectivity over 5-HT(2A) and 5-HT(2B). Among them, 6-methyl-N-[6-[(2-methyl-3-pyridinyl)oxy]-3-pyridinyl]1H-indole-3-carboxamide (8) exhibits the highest 5-HT(...

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Vydáno v:ACS Med Chem Lett
Hlavní autoři: Zeng, Fanxing, Nye, Jonathon A., Voll, Ronald J., Howell, Leonard, Goodman, Mark M.
Médium: Artigo
Jazyk:Inglês
Vydáno: American Chemical Society 2018
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC5846131/
https://ncbi.nlm.nih.gov/pubmed/29541358
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.7b00443
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