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Effects of adamantane alterations on soluble epoxide hydrolase inhibition potency, physical properties and metabolic stability

Adamantyl groups are widely used in medicinal chemistry. However, metabolism limits their usage. Herein, we report the first systematic study of adamantyl ureas and diureas bearing substituents in bridgehead positions of adamantane and/or spacers between urea groups and adamantane group, and tested...

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發表在:Bioorg Chem
Main Authors: Burmistrov, Vladimir, Morisseau, Christophe, Harris, Todd R., Butov, Gennady, Hammock, Bruce D.
格式: Artigo
語言:Inglês
出版: 2017
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在線閱讀:https://ncbi.nlm.nih.gov/pmc/articles/PMC5837815/
https://ncbi.nlm.nih.gov/pubmed/29310082
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bioorg.2017.12.024
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