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Effects of adamantane alterations on soluble epoxide hydrolase inhibition potency, physical properties and metabolic stability

Adamantyl groups are widely used in medicinal chemistry. However, metabolism limits their usage. Herein, we report the first systematic study of adamantyl ureas and diureas bearing substituents in bridgehead positions of adamantane and/or spacers between urea groups and adamantane group, and tested...

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Bibliografiske detaljer
Udgivet i:Bioorg Chem
Main Authors: Burmistrov, Vladimir, Morisseau, Christophe, Harris, Todd R., Butov, Gennady, Hammock, Bruce D.
Format: Artigo
Sprog:Inglês
Udgivet: 2017
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5837815/
https://ncbi.nlm.nih.gov/pubmed/29310082
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bioorg.2017.12.024
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